No | Name | Structure | IC50(nM) |
---|---|---|---|
1 | Cortistatin A | 17 | |
2 | SEL120-34A | 4 | |
3 | SenexinA | 280 | |
4 | SenexinB | 24–50 | |
5 | CCT251545 | 5 | |
6 | CCT251921 | 2.3 | |
7 | 3-Methyl-1H-pyrazolo(3,4-b)pyridine derivative | 4.4 | |
8 | 1,6-Naphthyridine derivative | 5.1 | |
9 | Isoquinoline derivative | 32.7 | |
10 | 3-Benzylindazole derivative | 53 | |
11 | 6-Azabenzothiophene derivative | 1.5 | |
12 | BRD6989 | \(\approx 500\) |